Intermediates

No. Name of Intermediates CAS No. API Name
1 (+/-)-3-(Carbamoylmethyl)-5-Methyl Hexanoic Acid (CMH) 181289-15-6 Pregabalin
2 R(-) -3- (Carbamoylmethyl)-5-Methyl Hexanoic Acid (RCMН) 181289-33-8 Pregabalin
3 Methyl 2-(4-(4-chlorobutanoyl)phenyl)-2-methylpropanoate 154477-54-0 Fexofenadine
4 alpha,alpha-Diphenyl-4-piperidinomethanol 115-46-8 Fexofenadine
5 Methyl 4-[4-[4-hydroxydiphenylmethyl)-1-piperidinyl] 1-oxobutyl]-2,2-dimethyl benzene acetate 154477-55-1 Fexofenadine
6 2-(2-hydroxyethyl)isoindoline-1,3-dione (Or) N-(2-Hydroxyethyl)phthalimide 3891-07-4 Amlodipine Besylate & Amlodipine Mesylate
7 Ethyl 4-(2-(1,3-dioxoisoindolin-2-yl)ethoxy)-3-oxobutanoate 88150-75-8 Amlodipine Besylate & Amlodipine Mesylate
8 phthaloyl Amlodipine 88150-62-3 Amlodipine Besylate & Amlodipine Mesylate
9 (R,S)-Amlodipine Base 88150-42-9 Amlodipine Besylate & Amlodipine Mesylate
10 2-(2-Thienyl)ethyl toluene-p-sulphonate 40412-06-4 clopidogrel bisulfate
11 (+) 2-(2-Chlorophenyl) glycine methyl ester (Tartrate Salt) 141109-15-1 clopidogrel bisulfate
12 S-(+)-Methyl-(2-chlorophenyl)[(2-(2-thienyl)amino] acetate hydrochloride 141109-19-5 clopidogrel bisulfate
13 2-(Aminomethyl)-1-ethylpyrrolidine 26116-12-1 Amisulpride
14 4-Amino-5-ethylsulfonyl-2-methoxybenzoic acid 71675-87-1 Amisulpride
15 (S)-2-(Aminomethyl)-1-ethylpyrrolidine 22795-99-9 Levosulpiride
16 1-ethyl-2-(nitromethylene)pyrrolidine 26171-04-0 Levosulpiride
17 Methyl-2-methoxy-5-sulfamoylbenzoate 33045-52-2 Levosulpiride
18 2-amino-5-methyl thiazole 7305-71-7 Meloxicam
19 4-hydroxy, 2-methyl-2h, 1,2-benzothiazine carboxylic acid isopropyl ester, 1,1-dioxide 118854-48-1 Meloxicam/Piroxicam
20 2H-Thieno-[2,3-e]-1,2- Thiazine-3-Carboxylic Acid, 6-Chloro-4-Hydroxy-2- Methyl Methylester-1,1- Dioxide 70415-50-8 Lornoxicam
21 2,3-Dichlorobenzoyl cyanide 77668-42-9 Lamotrigine
22 1,2,3,9-tetrahydro-4H-carbazol-4-one 15128-52-6 Carvedilol
23 4-(2,3-Ероxypropoxy) carbazole 51997-51-4 Carvedilol
24 2-(2-Methoxyphenoxy)ethylamine 1836-62-0 Carvedilol
25 2,4-Difluoro-alpha-(1h,1yl,1,2,4-Triazole) Acetophenone 86404-63-9 Fluconazole
26 (2,4-Difluorophenyl)-1-(1H-1,2,4-triazolyl)-2,3-epoxypropane methane sulfonate 86386-77-8 Fluconazole
27 5-chloro-2,4-di sulfamoyl aniline 121-30-2 Hydrochlorothiazide
28 p-Hydroxy Benzyl alcohol 623-05-2 Bisoprolol Fumarate
29 4-((2-isopropoxyethoxy) methyl)phenol 177034-57-0 Bisoprolol Fumarate
30 2-((4-((2-isopropoxyethoxy)methyl)phenoxy)methyl)oxirane 66722-57-4 Bisoprolol Fumarate
31 1,7'-Dimethyl-2'-propyl-2,5'-bibenzimidazole (BIM) 152628-02-9 Telmisartan
32 1-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazine 401566-79-8 Teneligliptin
33 4-(3'-Methylphenyl)amino-3-pyridinesulfonamide 72811-73-5 Torsemide
34 1-(2,3-Dichlorophenyl)Piperazine Hydrochloride 119532-26-2 Aripiprazole
35 Boc-(R)-3-amino-4-(2,4,5-trifluorophenyl)-butyric acid 486460-00-8 Sitagliptin
36 Alpha,alpha-dimethyl phenyl acetic acid 826-55-1 Bilastine / Fexofenadine
37 2-(piperidin-4-yl)-1H-benzo[d]imidazole 38385-95-4 Bilastine
38 2-ethoxyethyl 4-methylbenzenesulfonate 17178-11-9 Bilastine
39 2-[4-[1-(4,4-dimethyl-5H-oxazol-2-yl)-1-methylethyl]phenyl]ethyl 4-methylbenzenesulfonate 202189-76-2 Bilastine
40 Bromo-7-(2-butyn-1-yl)-3-methylxanthine 666816-98-4 Linagliptin
41 8-Bromo-7-but-2-ynyl-3-methyl-1-(4-methyl-quinazolin-2-ylmethyl)-3,7-dihydro-purine-2,6-dione 853029-57-9 Linagliptin
42 R-Boc-Amino-Piperidine 309956-78-3 Linagliptin
43 R-3-Aminopiperidine 2 HCl 334618-23-4 Linagliptin
44 2-Chloromethyl-3,4-dimethoxypyridinium chloride 72830-09-2 Pantoprazole
45 5-(Difluoromethoxy)-2-mercapto-1H-benzimidazole 97963-62-7 Pantoprazole
46 5-Difluoromethoxy-2-{[(3,4-dimethoxy-2-pyridinyl)methyl]thio}-1H-benzimidazole 102625-64-9 Pantoprazole
47 (4R,6R)-tert-Butyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxane-4-acetate 125971-94-0 Atorvastatin Calcium
48 4-Fluoro-alpha-(2-methyl-1-oxopropyl)-gamma-oxo-N,N-diphenylbenzene butaneamide 125971-96-2 Atorvastatin Calcium
49 tert-Butyl (4R,6R)-2-[[[6-(2,4-fluorophenyl)-5-isopropyl-3-phenyl-4-(phenylcarbamoyl)pyrrol-1-yl]ethyl]-2,2-dimethyl-1,3-dioxan-4-yl]acetate 125971-95-1 Atorvastatin Calcium
50 - - -
51 (S)-1-(Chloroacetyl)-2-pyrrolidine carboxamide 214398-99-9 Vildagliptin
52 3-Aminoadamantan-1-ol 702-82-9 Vildagliptin
53 4-(4-Aminophenyl)morpholine-3-one - Rivaroxaban
54 (S)-2-(Oxiran-2-ylmethyl)-1H-isoindole-1,3(2H)-dione 161596-47-0 Rivaroxaban